A K C G R O U P T K G R O U P C A M K G R O U P C K 1 G R ... T K G R O U P T K L G R O U P A T Y P I C A L I N H I B I T O R S B R O A D S P E C T R U M I N H I B I T O R S M I S

Kinase InhibitorsSTANDARDS I IMPURITIES I METABOLITES I INTERMEDIATES I LABELED

AKC GROUPCAMK GROUP CK1 GROUPCMGC GROUPSTE GROUP

TK GROUPTKL GROUPATYPICAL INHIB ITORSBROAD SPECTRUM INHIB ITORSMISCELLANEOUS

KinaseInhibitors

TorontoResearchChemicals,20MartinRossAvenue,NorthYork,ON,Canada,M3J2K8International:+1(416)665-9696,Fax:+1(416)665-4439

Email:[email protected]

ChemicalName CASNo. Cat.No.

α-AcetamidocinnamicAcid 5469-45-4 A150000

Genistein 446-72-0 G350000

1-(5-Isoquinolinesulfonyl)-2-methylpiperazineDihydrochloride 108930-17-2 I885000

1-(5-Isoquinolinesulfonyl)-3-methylpiperazineHydrochloride 141543-65-9 I885200

N-[2-(Methylamino)ethyl]-5-isoquinolinesulfonamideDihydrochloride 113276-94-1 M286200

rac-3-Octadecanamido-2-ethoxypropan-1-olPhosphocholine 112989-02-3 O234000

rac-3-Octadecanamido-2-Methoxypropan-1-olPhosphocholine 163702-19-0 O235000

Phloretin 60-82-2 P339000

D-erythro-Sphingosine(synthetic) 123-78-4 S681000

Zaprinast 37762-06-4 Z150000

rac3,4-DihydroxymandelicAcid 775-01-9 D453000

N-[2-(p-Bromocinnamylamino)ethyl]-5-IsoquinolineSulfonamide 127243-85-0 B682440

N-[2-(p-Cinnamylamino)ethyl]-5-isoquinoloneSulfonamide 130964-40-8 C442100

Tamoxifen 10540-29-1 T006000

3,4,5-TrimethoxybenzoicAcid8-(Diethylamino)octylEster,Hydrochloride 53464-72-5 T795650

Genistein-2’,3’,5’,6’-d4(Major) 187960-08-3 G350010

CaffeicAcidPhenethylEster 104594-70-9 C080050

CaffeicAcidDimethylEtherPhenethylEster 145551-14-0 C080010

1-Acetamido-4-cyano-3-methylisoquinoline 179985-52-5 A150525

N-[2-(p-Bromocinnamylamino)ethyl]-5-isoquinolineSulfonamide

Dihydrochloride

130964-39-5 B682445

N-Boc-erythro-sphingosine 116467-63-1 B667750

Fmoc-erythro-Sphingosine 56607-19-3 F667750

Azido-erythro-sphingosine 103348-49-8 A926500

2-Azido-1-pivaloylD-erythro-Sphingosine 114275-41-1 A925080

(2S,3R,4E)-2-Azido-3-(tert-butyldimethylsilyl)-1-pivaloyl-erythro-

sphingosine

114275-42-2 A822575

(2S,3R,4E)-2-Azido-3-(tert-butyldimethylsilyl)-erythro-sphingosine 114299-64-8 A822550

KinaseInhibitors



3-O-(tert-Butyldimethylsilyloxy)-erythro-sphingosine 137905-29-4 B691595

3-O-(tert-Butyldimethylsilyloxy)-2-Fmoc-erythro-sphingosine 149035-77-8 B691450

4,5,6,7-Tetrabromobenzimidazole 577779-57-8 T291150

Genistein-2’,6’-d2 315204-48-9 G350005

4-Benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione 327036-89-5 B285725

2,4-Dibenzyl-5-oxothiadiazolidine-3-thione 72966-20-2 D417960

Tamoxifen-d5 157698-32-3 T006077

KN-62 127191-97-3 K650000

4,5,6,7-Tetrabromo-1H-benzotriazole 17374-26-4 T291325

2-Azido-1,3-di-o-pivaloylD-erythro-Sphingosine A847625

H-1152Dihydrochloride 871543-07-6 H011520

1H-[1]-Benzazephe-2,5(3H,4H)-dione 16511-38-9 B186000

2-Amino-5-bromopyrazine-3-carboxylicAcidMethylEster 6966-01-4 A601863

3-Nitro-6-methylphenylguanidineNitrate 152460-08-7 N503755

N-(5-Amino-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine 152460-10-1 A618220

Staurosporin 62996-74-1 S685000

N-Boc-erythro-sphingosine-13C2,D2 B667752

D-erythro-Sphingosine-13C2,D2 S681002

TamoxifenN-Oxide 75504-34-6 T006095

N-Acetyl-4-aminosalicylicAcid 50-86-2 A168325

K252a 99533-80-9 K000500

N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamideDihydrochloride 1177141-67-1 A608851

N-(2-Aminoethyl)-5-isoquinolinesulfonamideHydrochloride 116970-50-4 A609001

N-(2-Chloro-6-methylphenyl)-2-[(6-chloro-2-methyl-4-pyrimidinyl)amino]-

5-thiazolecarboxamide

302964-08-5 C369290

(S)-2-Piperidineethanol 103639-57-2 P481955

(4R-cis)-6-Aminomethyl-2,2-dimethyl-1,3-dioxane-4-aceticAcidtert-Butyl

Ester

853881-01-3 A615950

N-(4-Pyridyl)-N’-(2,4,6-trichlorophenyl)urea 97627-27-5 P997000

DebromoHymenialdisine 75593-17-8 D208900

SU5402 215543-92-3 S688000

KinaseInhibitors



Paullone 142273-18-5 P207500

NU7441 503468-95-9 N925300

(R)-2-Piperidineethanol 68419-38-5 P481956

PamoicAcid-d10 1215327-33-5 P173502

AR-AO14418 487021-52-3 A765500

7-Azaoxindole 5654-97-7 A801725

4-Amino-5-(bromomethyl)-2-methylpyrimidineDihydrobromide 5423-98-3 A601820

BisindolylmaleimideVIIIAceticAcidSalt 138516-31-1 B448500

4-Amino-2-(methylthio)-5-pyrimidinecarboxylicAcidEthylEster 776-53-4 A618240

Balanol 63590-19-2 B115500

Curcumin 458-37-7 C838500

RuboxistaurinHydrochloride 169939-93-9 R701525

Curcumin-d6 1246833-26-0 C838502

Romidepsin 128517-07-7 R425060

3-(Methoxycarbonyl)phenylboronicAcid 99769-19-4 M261635

3-Methyl7-Azaoxindole 1330055-85-0 M288695

2-Hydroxymethyl-4-benzylmorpholine 40987-24-4 H946450

SB239063 193551-21-2 S154625

Selumetinib 606143-52-6 S254000

KN-93 139298-40-1 K653000

PD-184161 212631-67-9 P218100

6-Nitro-5-hydroxyNicotinicAcid 59288-43-6 N496200

1,4-Diaminoanthraquinone 128-95-0 D416080

2-(1-Naphthalenylcarbonyl)propanedinitrile 1236038-48-4 N368350

PamoicAcid 130-85-8 P173500

Genistein-4,6,2’,3’,5’,6’-d6

DiscontinuedSeeG350010

197657-74-2 G350002

AZD8055 1009298-09-2 A808130

Tamoxifen-13C6 1346606-38-9 T006002

2-Fluoro-3-iodo-5-methylpyridine 153034-78-7 F591970

KinaseInhibitors



1,2-Dichloro-4-methyl-3-nitro-5-(trifluoromethyl)benzene 115571-66-9 D435460

PHA767491DihydrochlorideSalt P294450

Vemurafenib 918504-65-1 V118500

BMS214662 195987-41-8 B596050

VX745 209410-46-8 V900500

Doramapimod 285983-48-4 D534250

Methyl5-Nitro-7-azaindole-2-carboxylate 952182-17-1 M323575

Talmapimod 309913-83-5 T005550

SB202190Hydrochloride 350228-36-3 S154500

VX-702 745833-23-2 V900250

Romidepsin-d8 R425062

PF-4708671 1255517-76-0 P294010

Vemurafenib-d5 1365986-90-8 V118502

O-tert-Butyl-dimethylsilylCurcumin 911292-36-9 B691020

Di-(tert-Butyl-dimethylsilyl)Curcumin 1134639-23-8 D428050

rac3,4-DihydroxymandelicAcid-d3 D453002

Ruboxistaurin-d6Hydrochloride 1794767-04-6 R701527

4-Amino-5-ethoxymethyl-2-methylpyrimidine 73-66-5 A609035

5-(Ethoxymethyl)-2-methyl-4-pyrimidinone 5423-97-2 E892470

PF-3644022 1276121-88-0 P293825

BisindolylmaleimideXIHydrochloride 145333-02-4 B448530

PF670462 950912-80-8 P293960

PF670462-d11 1794885-93-0 P293962

RWJ-67657 215303-72-3 R925200

2-[3-(Benzyloxy)phenyl]-2-methylpropionitrile 70120-08-0 B288205

3-Bromobenzene-1,2-diamine 1575-36-6 B680220

1-(5-Isoquinolinesulfonyl)-2-methyl-4-trityl-piperazine 1798013-99-6 I885010

3,3-Diethoxypropionitrile 2032-34-0 D442100

ML3403 549505-65-9 M425090

PF-3644022-d4 P293827

(R)-1-Aminopropan-2-ylcarbamicAcidtert-ButyEster 100927-10-4 A628140

KinaseInhibitors



TAK-960 1137868-52-0 T004940

BX-795 702675-74-9 B810550

CCT239065 1163719-51-4 C227950

PH-797804 586379-66-0 P399150

N,N-Di-(tert-Butyloxycarbonyl)Serotonin 361436-29-5 D428630

N-tert-ButyloxycarbonylSerotonin 53157-48-5 B693470

cis-7,10,13,16-DocosatetraenoicAcid 28874-58-0 D494510

ProcyanidinB2 29106-49-8 P755830

5-[2-(5-Nitro-2-furanyl)ethenyl]-2-furancarboxylicAcidMethylEster 24269-96-3 N493870

N-Demethyl-3,4-dihydroxytamoxifenHydrochloride

(Z,Emixture)

2125720-11-6 D231035

N-Demethyl-3,4-dihydroxytamoxifen-d3Hydrochloride

(Z,Emixture)

D231037

N-Demethyl-3-methoxy-4-hydroxytamoxifenHydrochloride

(E,Zmixture)

2125720-13-8 D231060

N-Demethyl-3-methoxy-4-hydroxytamoxifen-d3Hydrochloride

(Z,Emixture)

D231062

Rhein8-Glucoside 34298-86-7 R318520

7-Oxo-7H-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylicAcid 52029-86-4 O847425

3-Hydroxy-5,6,7,8-tetrahydro-10-oxa-8-aza-benzo[a]azulen-9-one 521937-07-5 H957795

(E)-3-(2,3,4,5-Tetrabromophenyl)acrylicAcid 934358-00-6 T291160

5-Methylindole 614-96-0 M313505

NSC177223 36707-00-3 N900270

BisindolylmaleimideIIIHydrochloride 683775-59-9 B448480

1-(5-Isoquinolinesulfonyl)-4-tert-butyloxycarbonyl-2-methylpiperazine 1796933-25-9 I885005

TAK-960-d3 T004942

(Oxazol-5-yl)ethylammoniumHydrochloride 317830-75-4 O858580

2-Fluoro-3-methoxybenzaldehyde 103438-88-6 F593270

L-O-Phosphoserine 407-41-0 P361200

L-O-Phosphoserine-13C315N P361202

3-Bromo-5,7-dichloro-pyrazolo[1,5-a]pyrimidine 114040-06-1 B684655

KinaseInhibitors



3-[1-(3-Hydroxypropyl)-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-1H-

pyrrole-2,5-dione

125313-60-2 H952665

3-[1-[3-(Hydroxy)propyl]-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-2,5-

furandioneAcetate

125314-97-8 H952670

2-[3-(1H-Indol-1-yl)propyl]-1H-isoindole-1,3(2H)-dione 150206-00-1 I633910

5-Chloro-2-nitroanisole 6627-53-8 C377695

SB202190 152121-30-7 S154495

4-DodecylbenzenesulfonicAcidPotassiumSalt 14564-74-0 D494560

CGK733 905973-89-9 P337400

AG-1295 71897-07-9 A425200

N-[5-[(4-Ethyl-1-piperazinyl)methyl]-2-pyridinyl]-5-fluoro-4-[4-fluoro-2-

methyl-1-(1-methylethyl)-1H-benzimidazol-6-yl]-2-pyrimidinamine

Methanesulfonate

1231930-82-7 E925710

Sotrastaurin 425637-18-9 S677600

2-Hydroxy-4’,5-diacetamido-biphenyl H825095

4-AcetamidophenylboronicAcid 101251-09-6 A158510

3-Chloro-2-pyrazinecarboxylicAcid 27398-39-6 C380420

3,5-Dichloro-2-pyrazinamine 873-42-7 D436135

GSK2606414 1337531-36-8 G797510

3-(Indolin-5-yl)-1-methyl-1H-pyrrolo[2,3-b]pyridin-4-amineHydrochloride I627250

GSK2606414-d3 G797512

Go6983 133053-19-7 G766495

(2S)-3-Phenyl-N1-[5,6,7,8-tetrahydro-2-(4-pyridinyl)[1]benzothieno[2,3-

d]pyrimidin-4-yl]-1,2-propanediamine

1438881-19-6 P336945

1,4-Dichlorophthalazine 4752-10-7 D436165

2-Amino-N-(2-chloro-6-methylphenyl)-5-thiazolecarboxamide 302964-24-5 A603910

1-Amino-2-propanol 78-96-6 A628135

B-[4-(Trifluoromethoxy)phenyl]boronicAcid 139301-27-2 T790910

α-[[(Phenylmethoxy)carbonyl]amino]-1H-benzotriazole-1-aceticAcid 124676-19-3 P335615

K252b 99570-78-2 K000505

N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamide 120615-25-0 A608850

KinaseInhibitors



rac-3-Hexadecanamido-2-ethoxypropan-1-olPhosphocholine

Monohydrate

H293000

N-[4-[(4-Chlorophenyl)methoxy]-2-pyridinyl]-2,6-difluoro-

benzeneacetamide

1415834-63-7 C380230

K252c 85753-43-1 K000510

(S)-(+)-2,2-Dimethyl-1,3-dioxolan-4-ylmethylp-Toluenesulfonate 23735-43-5 D469555

1-[4-[2-Dimethylamino)ethoxy]phenyl]-2-phenyl-1-butanone

Hydrochloride

94911-67-8 D461360

1-[4-[2-Dimethylamino)ethoxy]phenyl]-2-phenyl-1-butanone-d6

Hydrochloride

D461362

5-Amino-1-(1,1-dimethylethyl)-3-[(3-methylphenyl)methyl]-1H-pyrazole-

4-carbonitrile

A605035

GF109203X 133052-90-1 G368850

Ro31-8220Mesylate 138489-18-6 R637300

DorsomorphinDihydrochloride 1219168-18-9 D534910

4,5-DimethoxysalicylicAcid 5722-93-0 D461390

Sotrastaurin-d3 S677602

L-threo-Dihydrosphingosine 15639-50-6 D151740

N'-((4-(2-(Dimethylamino)ethoxy)phenyl)(phenyl)methylene)-4-

methylbenzenesulfonohydrazide

D461385

4-MethylbenzenesulfonicAcid2-[(4-

Hydroxyphenyl)phenylmethylene]hydrazide

147169-63-9 M226190

1,1,1-TrifluoromethanesulfonicAcid(E)-4-[1-[4-[2-

(Dimethylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]phenylEster

1370699-80-1 T790555

4-MethylbenzenesulfonicAcid2-[[4-[[(1,1-

Dimethylethyl)dimethylsilyl]oxy]phenyl]phenylmethylene]hydrazide

147169-61-7 M226210

(4-(2-(Dimethylamino)ethoxy)phenyl)(4-((4-(2-

(dimethylamino)ethoxy)phenyl)(phenyl)methyl)phenyl)methanone

D471135

4-((4-(2-(Dimethylamino)ethoxy)phenyl)(phenyl)methyl)-N-methoxy-N-

methylbenzamide

D471145

2-(4-((4-(4,4-Dimethyl-4,5-dihydrooxazol-2- D472730

KinaseInhibitors



yl)phenyl)(phenyl)methyl)phenoxy)-N,N-dimethylethanamine

(4-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)phenyl)(4-(2-

(dimethylamino)ethoxy)phenyl)(phenyl)methanol

D472735

2-(4-((4-(2-(Dimethylamino)ethoxy)phenyl)(phenyl)methyl)phenyl)-4,4-

dimethyloxazolidin-2-ol

D472745

4-(Dimethylaminoethoxy)benzophenone 51777-15-2 D472760

4-((4-(2-(Dimethylamino)ethoxy)phenyl)(phenyl)methyl)benzoicacid D472765

Imidazolo-oxindolePKRinhibitorC16

(PKRInhibitor)

608512-97-6 P572500

N-(tert-Butyl)-3-methylpicolinamide 32998-95-1 B693355

3-Amino-benzenemethanesulfonamide 344750-15-8 A591455

1-(3-Nitrophenyl)methanesulfonamide 110654-66-5 N493500

1,3-Dichloro-2-methyl-benzene 118-69-4 D435350

p-DodecylbenzenesulfonicAcidTriethanolamineSalt 3088-30-0 D493700

3-Phenylpropyne 10147-11-2 P336290

2-(((Benzyloxy)carbonyl)amino)-3-((diphenoxyphosphoryl)oxy)propanoic

AcidBenzylEster-13C,15N

B286757

N-(Benzyloxycarbonyl)serineBenzylEster 21209-51-8 B286770

N-(Benzyloxycarbonyl)serineBenzylEster-13C3,15N B286772

2-Bromothiazole-5-carboxylicAcid 54045-76-0 B688210

Ro31-8220Mesylate-d3 R637302

3-Amino-2-methoxycarbonylthiophene 22288-78-4 A612075

4-(1-(4-(2-Chloroethoxy)phenyl)-2-phenylbut-1-en-1-yl)-2-methoxyphenol

(E/ZMixture)

C367075

4-Bromo-2-hydroxypyridine 36953-37-4 B686020

3'-Bromopropiophenone 19829-31-3 B687240

CCT239065-d7 C227952

2-Aminobenzoxazole 4570-41-6 A591515

2-Fluoro-4-iodoaniline 29632-74-4 F591985

K02288 1431985-92-0 K000395

2-[4-[(1-(1,3-Benzodioxol-5-yl)-2-phenyl-1-buten-1-yl]phenoxy]-N,N- B276700

KinaseInhibitors



dimethylethanamineHydrochloride

(E/ZMixture)

5-[1-[4-(2-Chloroethoxy)phenyl]-2-phenyl-1-buten-1-yl]-1,3-benzodioxole

(E/ZMixture)

259149-68-3 C367120

1,3-Benzodioxol-5-yl[4-(2-chloroethoxy)phenyl]methanone 259149-65-0 B276705

WZ4003 1214265-58-3 W980000

CGP57380 522629-08-9 C583540

MK2InhibitorIII 724711-21-1 M424495

PHA767491 845714-00-3 P294445

YM201636 371942-69-7 Y100580

FR180204 865362-74-9 F763450

tert-Butyl(3-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)cyclohex-3-en-

1-yl)carbamate

1175298-09-5 T302650

(E/Z)-N,N-Didesmethyl-4-hydroxyTamoxifen-d5 D441122

TamoxifenCitrate 54965-24-1 T006090

cis-7,10,13,16-DocosatetraenoicAcidEthylEster 142828-41-9 D494730

cis-7,10,13,16-DocosatetraenoicAcidEthylEster-d5 D494732

4-[2-(Benzoyloxy)ethyl]-1,3-dihydro-2H-indol-2-one 139122-18-2 B208280

2-Methoxy-5-nitropyridine 5446-92-4 M265355

(20S)-Protopanaxadiol 30636-90-9 P838865

3,6-Diiodo-1H-indazole 319472-78-1 D454900

(2,2-Difluorocyclopropyl)methylamine 847926-81-2 D445435

WZ4003-d5 W980002

2-Hydroxy-4-methoxybenzaldehyde 673-22-3 H946010

4-Amino-5-ethoxymethyl-2-methylpyrimidineHydrobromide 115052-71-6 A609085

N-(1-Oxotetradecyl)-L-seryl-L-isoleucyl-L-tyrosyl-L-arginyl-L-arginylglycyl-

L-alanyl-L-arginyl-L-arginyl-L-tryptophyl-L-arginyl-L-lysyl-L-Leucine

863987-12-8 O870410

3-Bromo-4-fluoro-benzoicAcidEthylEster 23233-33-2 B683775

KT5823 126643-37-6 K660350

CX-4945 1009820-21-6 C858600

1-Methoxy-2-propanol 107-98-2 M265005

KinaseInhibitors



ChelerythrineChloride 3895-92-9 C291880

Genistein4'-β-D-glucopyranoside 152-95-4 G349975

3-Bromo-6-chloroimidazo[1,2-b]pyridazine 13526-66-4 B682330

PH-797804-d5 P399152

3-(Bromomethyl)toluene 620-13-3 B687610

Rp-CyclicAMPS 151837-09-1 R700920

(S)-(-)-PH-797804 1358027-80-1 P399155

Genistein7-SulfateSodiumSalt G350045

4-Chlorophthalazin-1-amine 13580-86-4 C380555

Rp-8-CPT-CyclicAMP(SodiumSalt) 221905-35-7 R700925

2-Amino-3-carboethoxy-4-(3-methylphenyl)thiophene 255713-71-4 A612160

BisindolylmaleimideXHydrochloride 145317-11-9 B448525

2,4-Dichloro-5-trifluoromethylpyrimidine 3932-97-6 D436635

KD025 911417-87-3 K145600

KU-60019 925701-46-8 K660435

1-O-Hexadecyl-2-O-methylglycerol 84337-41-7 H290985

Ethyl6-Cyano-1H-indole-2-carboxylate 104291-81-8 E907940

Di-O-glycinoylcurcuminDihydrochloride 1322544-82-0 D455700

Di-O-glycinoylcurcumin-d6Dihydrochloride D455702

Di-O-cysteinyl-glycinoylCurcumin90% 1042019-87-3 D455600

Di-O-cysteinyl-glycinoylCurcumin-d6 D455602

N,N'-Diphthaloyl-L-cystine 29588-96-3 D492235

1-O-Hexadecyl-2-O-methylglycerol-d5 H290987

rac-Balanol 167937-47-5 B115505

rac-syn-Balanol 167937-50-0 B115510

2-(1-Piperidino)aniline 39643-31-7 P481935

5,8-Diamino-1,4-dihydroxyanthraquinone 16517-70-7 D416155

Pim-1Inhibitor2 477845-12-8 P446710

3'-Methoxy-4',5,7-trihydroxyisoflavone 36190-95-1 M269675

BB-9000 947533-21-3 B119135

2-(2-Chloropyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 724726-05-0 C380645

KinaseInhibitors



2-Chloro-4-cyanopyridine 33252-30-1 C380665

2-Bromo-1-(2-chloropyridin-4-yl)ethanoneHydrobromide 569667-89-6 B682540

2-Acetamido-5-chloroisonicotinicAcid 944390-08-3 A150100

2-Acetylamino-4-methylpyridine 5327-32-2 A168500

AZD2932 883986-34-3 A808170

3-Chloro-2,5-difluoropyridine 851179-00-5 C368285

1-Benzyl-4-methylpiperidin-3-one 32018-96-5 B287190

N-Methoxy-N-methylbenzamide 6919-61-5 M265920

N-(5-Amino-2-methylphenyl)guanadineNitrate A617065

N,N’-Di-Boc-S-di(trityl)-di-O-cysteinyl-glycinoylCurcumin D420025

tert-Butyl5-Amino-1H-indazole-1-carboxylate 129488-10-4 B689775

LeucicAcid 498-36-2 L330080

3-(Diethylboryl)pyridine 89878-14-8 D442040

BisindolylmaleimideXIHydrochloride-d6 B448532

Methyl3-(Bromomethyl)benzoate 1129-28-8 M294015

1,3-Benzothiazol-2-ylacetonitrile 56278-50-3 B206655

6-Bromo-3-(1-methyl-1H-pyrazol-4-yl)-5-(3S)-3-piperidinylpyrazolo[1,5-

a]pyrimidin-7-amine

891494-64-7 B685536

XL228 898280-07-4 X746000

MGCD516 1123837-84-2 M340970

Hypothemycin 76958-67-3 H998480

2-Chloro-6-iodopyridine 258506-66-0 C368580

tert-ButylN-(4-Amino-1-methylcyclohexyl)carbamate 1254058-26-8 B693140

tert-ButylN-(4-Amino-1-methylcyclohexyl)carbamate-d3 B693142

OD36 1638644-62-8 O241600

OD38 1638644-63-9 O241605

Trans-1,2-cyclohexanedicarboxylicAnhydride 14166-21-3 C987290

6-Methoxyimidazo[1,2-a]pyridine 955376-51-9 M268505

(±)-1,2-Diphenyl-1-[4-[2-(dimethylamino)ethoxy]phenyl]butan-1-ol 748-97-0 D489850

PurvalanolB 212844-54-7 P840360

NSC693868 40254-90-8 N900555

KinaseInhibitors



(±)-1,2-Diphenyl-1-[4-[2-(dimethylamino)ethoxy]phenyl]butan-1-ol-d5 D489852

α-[4-(2-Dimethylaminoethoxy)phenyl]stilbene 19957-51-8 D471495

α-[4-(2-Dimethylaminoethoxy)phenyl]stilbene-d6 D471497

CDK1/2InhibitorIII 443798-55-8 C228110

2-[4-(1,2-Diphenyl-1-propenyl)phenoxy]-N,N-dimethylethanamine(E/Z

Mixture)

197251-11-9 D492270

2-[4-(1,2-Diphenyl-1-propenyl)phenoxy]-N,N-dimethylethanamine-d6

(E/ZMixture)

D492272

(±)-1,2-Diphenyl-1-[2-[2-(dimethylamino)ethoxy]phenyl]butan-1-ol D489855

(±)-1,2-Diphenyl-1-[2-[2-(dimethylamino)ethoxy]phenyl]butan-1-ol-d5 D489857

AktInhibitorXI 902779-59-3 A450500

4-[(2,4-Dichloro-5-methoxyphenyl)amino]-7-hydroxy-6-methoxy-3-

quinolinecarbonitrile

1460227-29-5 D435345

3-[4-Aminosulfonyl)phenyl]-2-propenoicAcid 147723-92-0 A629520

tert-Butyl2,6-diazaspiro[3.4]octane-2-carboxylate 885270-84-8 B694015

ZincCyanide 557-21-1 Z439500

N-Desdimethylaminoethyl-N-methylNitro-N'-desacryloylOsimertinib 1820891-36-8 D291260

4-Amino-2-chlorobenzamide 211374-81-1 A609310

4,6-Dichloro-3-fluoro-1H-pyrazolo[3,4-d]pyrimidine D434455

1-(3-Aminopropyl)imidazole 5036-48-6 A608805

ortho-TopolinRiboside-5‘-MonophosphateSodiumSalt 1343484-40-1 T540295

Oxazol-5-ylboronicAcid 808126-65-0 O858585

3-(4-Methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)benzonitrile 641571-12-2 M313025

2-BromobenzylBromide 3433-80-5 B679975

6-FluoresceinIsothiocyanate 3326-31-6 F485710

N-Acetyl-4-aminosalicylicAcid-d3 A168327

2,3-Dichloro-6-nitrobenzaldehyde 75618-41-6 D436955

1,1,1-Trifluoro-methanesulfonicAcid3-[[(1,1-

Dimethylethoxy)carbonyl]amino]-1-cyclohexen-1-ylEster

1803033-60-4 T779050

1,1,1-Trifluoro-methanesulfonicAcid5-[[(1,1-

Dimethylethoxy)carbonyl]amino]-1-cyclohexen-1-ylEster

1803033-59-1 T779055

KinaseInhibitors



2-Amino-3-ethynylpyrazine 1005349-13-2 A608290

2-Amino-3-hydroxypyrazine 43029-19-2 A612480

2-(N,N-BisBOC-Amino)pyrimidine-5-boronicAcid,PinacolEster 1190423-36-9 B404943

4-(4-BOC-Piperazino)phenylboronicacid 457613-78-4 B661998

Methyl3-Amino-6-chloropyrazine-2-carboxylate 1458-03-3 M328775

Vps34-IN-1 1383716-33-3 V785030

GSK2141795C 1047634-65-0 G797425

CellSheetMigrationInhibitor,Locostatin 133812-16-5 C256503

Pseudohypericin 55954-61-5 P839563

TX-1123 157397-06-3 T700575

BenzylSelenocyanate 4671-93-6 B289303

kbNB142-70 1233533-04-4 N381305

UCN-02 121569-61-7 U130603

Rp-8-Br-PET-cyclicGMPSSodiumSalt 185246-32-6 R700933

BML-275 866405-64-3 B595893

AktInhibitorIV 681281-88-9 A450505

ST638 107761-24-0 S687210

Palmitoyl-DL-carnitinechloride 6865-14-1 P163658

Wighteone 51225-30-0 W499205

Isowighteone 68436-47-5 I918230

Lupiwighteone 104691-86-3 L478020

CRT5 1034297-58-9 C782015

FRAX597 1286739-19-2 F763805

4-[1-(6-Quinolinylmethyl)-1H-1,2,3-triazolo[4,5-b]pyrazin-6-yl]-1H-

pyrazole-1-ethanol

956905-27-4 Q750035

N-[3-[[5-Cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-

pyrimidinyl]amino]propyl]cyclobutanecarboxamide

1190378-57-4 C986950

4-Methoxy-3-(2S)-2-morpholinyl-benzonitrileHydrochloride 881919-99-9 M330008

2-Chloro-6-morpholinopyran-4-one 119671-47-5 C379145

CGP60474 164658-13-3 C291780

HTH01-015 1613724-42-7 H671505

KinaseInhibitors



OTS514 1338540-63-8 O712950

5-Fluoro-AMB 1801552-03-3 F587305

LDC4297 1453834-21-3 L367665

AV412 451493-31-5 A794725

Methyl2-Amino-4-benzyloxy-5-methoxybenzoate 61032-42-6 M292985

4-Dodecylphenyl-13C61-SodiumSulfonate D494569

RheinMethylate 6155-37-9 R318525

RheinMethylate2,3,4,6-Tetraacetateβ-D-Glucopyranose R318530

RheinMethylate3-(2,3,4,6-Tetraacetateβ-D-Glucopyranose) R318535

rac-Talmapimod 309915-13-7 T005540

3-Iodo-3H-pyrazolo[3,4-d]pyrimidin-4-amine 151266-23-8 I736005

4-Amino-2-chlorobenzeneaceticAcid 50712-59-9 A603915

N161 141774-20-1 N185500

N-[3-[3-(2-Amino-2-oxoethyl)-1H-indol-1-yl]propyl]-carbamicAcid1,1-

DimethylethylEster

1024583-85-4 A616315

5-Ethoxychelerythrine 79559-55-0 E891745

APY29 1216665-49-4 A735420

Dasatinibmonohydrate 863127-77-9 D193638

1H-Pyrazole-4-boronicAcid 763120-58-7 P842210

2-Cyanoethylalsterpaullone 852527-97-0 C979580

2-Amino-1-phenyl-1,3-propanediol 55057-81-3 A627345

7-Ethyl-1H-indole-2,3-dione 79183-65-6 E702963

BX-795Hydrochloride 1472611-45-2 B810603

AMG548 864249-60-5 A614420

AminoguanidineHydrochloride 1937-19-5 A609863

AV412 451492-95-8 A794728

AZ3146 1124329-14-1 A808218

BisindolylmaleimideII 137592-45-1 B448535

CE3F4 143703-25-7 C228805

Centrinone 1798871-30-3 C256613

CGP52411 145915-58-8 C583570

KinaseInhibitors



CHIR99021 252917-06-9 C292155

CMPD-1 41179-33-3 C594953

Dihydrosphingosine 3102-56-5 D151745

HS38 1030203-81-6 H671503

KN93Phosphate 1188890-41-6 K653505

Necrosulfonamide 1360614-48-7 N388605

SB203580Hydrochloride 869185-85-3 S155058

U0124 108923-79-1 U850345

Akt-I-1 473382-39-7 A450508

2-((4-(2-Fluorophenoxy)phenyl)amino)acetonitrile 1415932-47-6 F594332

AS1940477Hydrobromide 1404189-10-1 A790093

4-Methyl-N-[4-methyl-3-[[4-(3-pyridinyl)-2-

pyrimidinyl]amino]phenyl]benzamideMethaneSulpfonate

M321305

4-(4-(3-(4-Chloro-3-(trifluoromethyl)phenyl)ureido)-3-

fluorophenoxy)picolinicAcid

1187945-05-6 C596470

3,7-Dihydro-3-[3-(3-hydroxyphenyl)-2-propyn-1-yl]-1,7-dimethyl-8-

(methylsulfonyl)-1H-purine-2,6-dione

2093393-05-4 D679023

M-3814 1637542-33-6 M199265

[1-(Ethylamino)cyclohexyl]methanol 852108-26-0 E900118

O-tert-Butyl-dimethylsilylCurcumin-d6 B691022

Di-(tert-Butyl-dimethylsilyl)Curcumin-d6 D428052

CC-671 1618658-88-0 C227915

4-Hydroxy-β-CarboxyTamoxifenO-Glucuronide T006055

4-Hydroxy-β-CarboxyTamoxifenN-β-D-Glucuronide H805270

4-Hydroxy-TamoxifenAcyl-glucuronide H805275

IvacaftorAcyl-Glucuronide I940630

N'-[3-[5-(2-Amino-4-pyrimidinyl)-2-(1,1-dimethylethyl)-4-thiazolyl]-2-

fluorophenyl]-N-ethyl-N-methylsulfamide

1638772-61-8 A634595

(2,6-Dichlorophenyl)methanamine 6575-27-5 D437840

(2-Methyl-1H-indol-5-yl)methylamine 36798-25-1 M313478

Ethyl2-Amino-4-(3,4-dimethylphenyl)thiophene-3-carboxylate 307511-65-5 B433788

KinaseInhibitors



6-Amino-2,2-dimethyl-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one 1002726-62-6 A634765

Pyrazolo[1,5-a]pyrimidine 274-71-5 P846520

TCKHNS11 1431540-99-6 T127788

AZD6738 1352226-88-0 A965423

1,2-Dihydro-2,5-diphenyl-3H-pyrazol-3-one 6632-05-9 D452723

2-Methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)quinoline 1022090-86-3 M332360

rac-1,2-Dioctanoyl-3-Chloropropanediol 95610-54-1 D481180

rac-1,2-Dioctanoyl-3-Chloropropanediol-d5 D481182

rac-1,2-Dioctanoyl-3-Chloropropanediol-13C3 D481183

6,8-Dihydro-8-(methylthio)-7H-pyrrolo[2,3-g]benzothiazol-7-one 222036-26-2 D453653

Fasudil 103745-39-7 F150023

2-Aminopurine 452-06-2 A628918

1-(2-Thiazolylazo)-2-naphthol 1147-56-4 T779315

D-Erythro-SphingosineSulfate 56607-20-6 S681505

6,8-Dihydro-7H-pyrrolo[2,3-g]benzothiazol-7-one 222036-27-3 D453658

GSK'872 1346546-69-7 G797855

Methyl5-Iodo-1H-indazole-3-carboxylate 1079-47-6 M322705

4-{[2-(Thiophen-2-yl)ethyl]sulfamoyl}benzoicAcid 1031130-62-7 B586783

4-(3-Aminophenyl)-3-morpholinone 1082495-22-4 A638210

Tamoxifen(1.0mg/mLinMethanol) 10540-29-1 KIT8260

Methyl(1-methylindolyl)-3-glyoxylate 151490-40-3 M336200

8-[(Hexahydro-1H-1,4-diazepin-1-yl)sulfonyl]isoquinoline 166895-76-7 H296915

5-[(Hexahydro-4-hydroxy-1H-1,4-diazepin-1-yl)sulfonyl]isoquinoline 1350827-92-7 H296920

6-Amino-5-methyl-3-pyridinecarboxylicAcidMethylEster 1184913-79-8 M335018

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