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Equestrian Canada Drug Classification Scheme This Classification Scheme does not constitute a Prohibited List of banned substances not allowed in horses. Rather, it is designed to allow a hearing panel, after an equine medication violation has been determined, to determine the most appropriate sanction. The drugs, medications and types of substances listed under each Class are not exhaustive. The list in each Class provides examples of drugs, medications and types of substances with similar effects on a horse or that are considered equivalently serious when detected in a horse participating in an EC sanctioned competition. Sanctions will be imposed on a Class by Class basis. Class 1: - Substances which have no place in performing horses. Many of these compounds do not have legitimate medical uses in horses, and the remaining compounds would only be used for severely debilitated animals. Abuse of these compounds is of serious ethical (and many cases, legal) concern. - Most of these compounds are included in Schedules 1 and 3 of the Canadian Controlled Drugs and Substances Act (CDSA) - Examples of Class 1 drugs: o Opioids such as fentanyl, morpine, heroin and codeine o Cocaine o Amphetamine and its derivatives listed in Schedule 3 of the CDSA o Methylphenidate (Ritalin) o Methaqualone Class 2: - These compounds are not appropriate for use around the time of performance. Inappropriate use may alter the horse’s behaviour and ability to perform; medical use of these compounds indicates health status incompatible with athletic competition. - Benzodiazepines - Barbiturates - Beta-adrenergic agonists not approved for use in horses - Local anesthetics - Erythropoietin, darbepoietin - Non-depolarizing muscle relaxants (e.g., pancuronium, vecuronium) - Tricyclic antidepressants - Monoamine oxidase inhibitors (antidepressants) - Antipsychotic drugs including most phenothiazines (so fluphenazine is included here but acepromazine is not) - Ketamine - Guaifenesin

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Page 1: Equestrian Canada Drug Classification Scheme

Equestrian Canada Drug Classification Scheme

This Classification Scheme does not constitute a Prohibited List of banned substances not allowed in horses. Rather, it is designed to allow a hearing panel, after an equine medication violation has been determined, to determine the most appropriate sanction. The drugs, medications and types of substances listed under each Class are not exhaustive. The list in each Class provides examples of drugs, medications and types of substances with similar effects on a horse or that are considered equivalently serious when detected in a horse participating in an EC sanctioned competition. Sanctions will be imposed on a Class by Class basis.

Class 1:

- Substances which have no place in performing horses. Many of these compounds do not have legitimate medical uses in horses, and the remaining compounds would only be used for severely debilitated animals. Abuse of these compounds is of serious ethical (and many cases, legal) concern.

- Most of these compounds are included in Schedules 1 and 3 of the Canadian Controlled Drugs and Substances Act (CDSA)

- Examples of Class 1 drugs: o Opioids such as fentanyl, morpine, heroin and codeine o Cocaine o Amphetamine and its derivatives listed in Schedule 3 of the CDSA o Methylphenidate (Ritalin) o Methaqualone

Class 2: - These compounds are not appropriate for use around the time of performance. Inappropriate use may alter

the horse’s behaviour and ability to perform; medical use of these compounds indicates health status incompatible with athletic competition.

- Benzodiazepines - Barbiturates - Beta-adrenergic agonists not approved for use in horses - Local anesthetics - Erythropoietin, darbepoietin - Non-depolarizing muscle relaxants (e.g., pancuronium, vecuronium) - Tricyclic antidepressants - Monoamine oxidase inhibitors (antidepressants) - Antipsychotic drugs including most phenothiazines (so fluphenazine is included here but acepromazine is

not) - Ketamine - Guaifenesin

Page 2: Equestrian Canada Drug Classification Scheme

Class 3: - Unapproved NSAIDs - Cases where multiple approved NSAIDs are detected - Anabolic steroids - Drugs used for standing sedation (butorphanol, acepromazine, detomidine, romifidine, xylazine) - Alpha-2 adrenergic agonist reversal agents (yohimbine, tolazoline) - Anticholinergics (atropine, glycopyrrolate, hyoscine/scopolamine and derivatives) - Ephedrine - Caffeine - Cardiovascular drugs

o ACE inhibitors o Phosphodiesterase inhibitors (including sildenafil) o Calcium channel blockers o Beta-blockers o Digoxin, digitoxin

- Antihistamines including hydroxyzine - Non-barbiturate anti-convulsants - Ergoloid mesylates and ergot alkaloids (current testing does not cover pergolide mesylate)

Class 4: - NSAIDs approved for use in horses in Canada, detected alone (where event-specific rules prohibit such

use) - Diuretics (including thiazide diuretics, acetazolamide, furosemide and other loop diuretics) - Muscle relaxants - Dembrexine - Corticosteroids - Isoxsuprine - Parasympathomimetics including bethanechol - DMSO - Altrenogest - Medroxyprogesterone

Class 5: - Mast cell stabilizers (Cromolyn, nedocromil) - Proton pump inhibitors except omeprazole - H2 antagonists except ranitidine and cimetidine - Misoprostol - Anticoagulants - Does NOT include polyethylene glycol

Page 3: Equestrian Canada Drug Classification Scheme

The drugs and medications listed below are not exhaustive. The list merely represents examples of the more common drugs and medications associated with each Class.

Drug Alternative names/examples Class Alfentanil Alfenta 1 Amphetamine 1 Amphetamine derivatives listed in the Canadian Controlled Drugs and Substances Act MDMA (Ecstasy), methamphetamine 1 Anileridine Leritine 1 Apomorpnine 1 Benzylpiperazine (BZP) 1 Carfentanil 1 Cathinone Khat, kat, qat, quat, chat, catha, Abyssinian tea, African tea 1 Cocaine 1 Codeine 1 Dextromoramide Palfium, Narcolo 1 Diamorphine 1 Dihydrocodeine Parcodin 1 Donepezil Aricept 1 Ethylmorphine Dionin 1 Etorphine M99 1 Exogenous endorphins 1 Exogenous enkephalins 1 Fentanyl Sublimaze, Duragesic 1 Heroin 1

Page 4: Equestrian Canada Drug Classification Scheme

Hydrocodone (dihydrocodeinone) Hycodan 1 Hydromorphone Dilaudid 1 Hydroxyamphetamine Paradrine 1 Levomethorphan 1 Levorphanol Levo-Dremoran 1 Lofentanil 1 Mazindol Sanorex 1 Meperidine Demerol 1 Mephentermine 1 Metaraminol Aramine 1 Methadone Dolophine 1 Methamphetamine Desoxyn 1 Methaqualone Quaalude 1 Methcathinone 1 Methylphenidate Ritalin 1 Metopon (Methyldihydromorphinone) 1 Morphine 1 Nikethamide Coramine 1 Oxycodone Percodan 1 Oxymorphone Numorphan 1 Pemoline Cylert 1 Pentazocine Talwin 1 Pentylenetetrazole Metrazol, Nioric 1 Phenazocine Narphen 1 Phencyclidine (PCP) Sernylan 1

Page 5: Equestrian Canada Drug Classification Scheme

Phendimetrazine Bontril 1 Picrotoxin 1 Piritramide 1 Remifentanil Ultiva 1 Strychnine 1 Sufentanil Sufenta 1 Acecarbromal 2 Acetophenazine Tindal 2 Adinazolam 2 Alcuronium Alloferin 2 Alphaprodine Nisentil 2 Alpidem Anaxyl 2 Alprazolam Xanax 2 Althesin Saffan 2 Amisulpride Solian 2 Amitriptyline Elavil 2 Amobarbital Amytal 2 Amoxapine Asendin 2 Amperozide 2 Anilopam Anisine 2 Aprobarbital Alurate 2 Articaine Septocaine, ultracaine 2 Atomoxetine Strattera 2 Atracurium Tracrium 2 Azacylonol Frenque 2

Page 6: Equestrian Canada Drug Classification Scheme

Azaperone Stresnil 2 Barbital Veronal 2 Barbiturates 2 Bemegride Megimide 2 Benoxinate Dorsacaine 2 Benperidol 2 Bentazepam Tiadipona 2 Benzactizine Deprol, Bronchodiletten 2 Benzocaine 2 Benzoctamine 2 Benzodiazepines 2 Benzphetamine Didrex 2 Benztropine Cogentin 2 Biriperone 2 Bromazepam Lexotan, Lectopam 2 Bromisovalum Diffucord 2 Bromocriptine Parlodel 2 Bromperidol Bromidol 2 Brotizolam Brotocol 2 Bupivacaine Marcaine 2 Buprenorphine Temgesic 2 Bupropion Wellbutrin 2 Buspirone Buspar 2 Butabarbital (Secbutobarbitone) Butacaps, butasol 2 Butacaine Butyn 2

Page 7: Equestrian Canada Drug Classification Scheme

Butalbital (Talbutal) Florinal 2 Butanilicaine Hostacain 2 Butaperazine Repoise 2 Butoctamide 2 Captodiame Covatine 2 Carbidopa & levodopa Sinemet 2 Carbromol Mifudorm 2 Carisoprodol Rela, Soma 2 Carmazepam Paxor 2 Carphenazine Proketazine 2 Carpipramine Prazinil 2 Carticaine Septocaine, ultracaine 2 Chloral betaine Beta-chlor 2 Chloral hydrate 2 Chloraldehyde (Chloral) 2 Chloralose (Alpha-chloralose) 2 Chlorazepate Tranxene 2 Chlordiazepoxide Librium 2 Chlorhexidol 2 Chlormezanone Trancopal 2 Chloroform 2 Chloroprocaine Nesacaine 2 Chlorproethazine Newiplege 2 Chlorpromazine Thorazine, Largactil 2 Chlorprothixene Taractan 2

Page 8: Equestrian Canada Drug Classification Scheme

Cinchocaine Nupercaine 2 Citalopram Celexa 2 Clibucaine 2 Clobazam Urbanyl 2 Clocapramine 2 Clomethiazole 2 Clomipramine Clomicalm, Anafranil 2 Clonazepam Klonopin 2 Clormecaine 2 Clothiapine Entermin 2 Clotiazepam Trecalmo, Rize 2 Cloxazolam Enadel, Sepazon, Tolestan 2 Clozapine Clozaril, Leponex 2 Conorphone 2 Corticaine Ultracain 2 Crotetamide 2 Cyamemazine 2 Cyclobarbital Phanodorm 2 Darbepoetin Aranesp 2 Decamethonium Syncurine 2 Demoxepam 2 Desipramine Norpromine 2 Dezocine Dalgan 2 Diazepam Valium 2 Dibucaine Nupercainal, Cinchocaine 2

Page 9: Equestrian Canada Drug Classification Scheme

Dichloralphenazone Febenol, Isocom 2 Diethylpropion Tepanil 2 Diethylthiambutene Themalon 2 Dilorazepam Briantum 2 Dimethisoquin 2 Diprenorphine M50/50 2 Dixyrazine Esucos 2 Dopamine Inotropin 2 Doxacurium Nuromax 2 Doxapram Dopram 2 Doxefazepam Doxans 2 Doxepin Adapin, Sinequan 2 Droperidol 2 Enciprazine 2 Epibatidine 2 Estazolam 2 Ethamivan 2 Ethanol 2 Ethclorvynol Placidyl 2 Ethinamate Valmid 2 Ethopropazine Parsidol 2 Ethylisobutrazine Diquel 2 Etidocaine Duranest 2 Etifoxin Stresam 2 Etizolam Depas, Pasaden 2

Page 10: Equestrian Canada Drug Classification Scheme

Etodroxizine Indunox 2 Etomidate 2 Exogenous erythropoietin (EPO) Epogen 2 Fenarbamate Tymium 2 Fenfluramine Pondimin 2 Fluanisone Sedalande 2 Fludiazepam Erispam 2 Flunitrazepam Rohypnol, Narcozep, Hypnodorm 2 Fluopromazine Psyquil 2 Fluoresone Caducid 2 Fluoxetine Prozac 2 Flupenthixol Depixol, Fluanxol 2 Fluphenazine Prolixin, Modecate 2 Flurazepam Dalmane 2 Fluspirilene Imap, Redeptin 2 Flutoprazepam Restas 2 Fluvoxamine Dumirox, Faverin 2 Galantamine Reminyl 2 Gallamine 2 Gamma amino butyric acid GABA 2 Gepirone 2 Glutethimide Doriden 2 Halazepam Paxipam 2 Haloperidol Haldol 2 Haloxaazolam Somelin 2

Page 11: Equestrian Canada Drug Classification Scheme

Hemoglobin glutamers Oxyglobin, Hemopure 2 Hexafluorenium Myalexen 2 Hexobarbital Evipal 2 Hexylcaine 2 Homophenazine Pelvichthol 2 hydroxy-gamma butyric acid Hydroxy-GABA 2 Ibomal Noctal 2 Imipramine Tofranil 2 Injectable Magnesium 2 Isapirone 2 Isocarboxazid Marplan 2 Isomethadone 2 Isoproterenol Isoprel 2 Ketamine Ketaset 2 Ketazolam Anxon 2 Lenperone Elanone-V 2 Lidocaine Xylocaine 2 Lithium 2 Lobeline 2 Loflazepate (ethyl-) Victan 2 Loperimide Imodium 2 Loprazolam Dormont 2 Lorazepam Ativan 2 Lormetazepam Noctamid 2 Loxapine Laxitane 2

Page 12: Equestrian Canada Drug Classification Scheme

Maprotiline Ludiomil 2 Mebutamate Axiten 2 Meclofenoxate Lucidril 2 Medazepam Nobrium 2 Melperone Eunerpan 2 Memantine Namenda 2 Meparfynol Oblivon 2 Mepazine Pacatal 2 Mephenoxalone Control 2 Mephenytoin Mesantoin 2 Mephobarbital (Methylphenobarbital) Mebaral 2 Mepivacaine Carbocaine V 2 Meprobamate Equanil 2 Mesoridazine Serentil 2 Metaclazepam Talis 2 Metazocine 2 Metharbital Gemonil 2 Methohexital Brevital 2 Methotrimeprazine Levoprome 2 Methylprylon Noludar 2 Metocurine Metubine 2 Metomidate Hypnodil 2 Mexazolam Melex 2 Midazolam Versed 2 Mirtazepine Remeron 2

Page 13: Equestrian Canada Drug Classification Scheme

Mivacurium Mivacron 2 Modafinil Provigil 2 Molindone Moban 2 Moperone Luvatren 2 Mosaprimine 2 Nalbuphine Nubain 2 Nalorphine Nalline 2 Nefazodone Serzone 2 Nimetazepam Erimin 2 Nitrazepam Mogadon 2 Nordiazepam Calmday 2 Norepinephrine 2 Nortriptyline Aventyl 2 Olanzepine Zyprexa 2 Oxazepam Serax 2 Oxazolam Serenal 2 Oxyperitine Forit 2 Pancuronium Pavulon 2 Paraldehyde Paral 2 Paroxetine Paxil 2 Penfluridol Cyperon 2 Pentobarbital Nembutal 2 Perazine Taxilan 2 Perfluorocarbons 2 Perfluorodecahydronophthalene 2

Page 14: Equestrian Canada Drug Classification Scheme

Perfluorodecolin 2 Perfluorooctylbromide 2 Perfluorotripopylamine 2 Periciazine Alodept 2 Perlapine Hypnodin 2 Perphenazine Trilafon 2 Phenaglycodol Acalo 2 Phenelzine Nardil 2 Phenobarbital Luminal 2 Phentermine Iomamin 2 Piminodine Alovodine, Cimadon 2 Pimozide Orap 2 Pinazepam Domar 2 Pipamperone Dipiperon 2 Pipecuronium Arduan 2 Pipequaline 2 Piperacetazine Psymode, Quide 2 Piperocaine Metycaine 2 Pipotiazine Lonseren 2 Pipradol Dataril 2 Piquindone 2 Prazepam Verstran, Centrax 2 Prilocaine Citanest 2 Prochlorperazine Darbazine, Compazine 2 Propanidid 2

Page 15: Equestrian Canada Drug Classification Scheme

Proparacaine 2 Propiomazine Largon 2 Propionylpromazine Tranvet 2 Propiram 2 Propofol Propoflo, Rapinovet 2 Propoxycaine Ravocaine 2 Prothipendyl Dominal 2 Protriptyline Concordin, Triptil 2 Proxibarbital Axeen 2 Pyrithiyldione Hybersulfan 2 Quazipam Doral 2 Quetiapine Seroquel 2 Racemethorphan 2 Racemorphan 2 Raclopride 2 Ractopamine Paylean 2 Remoxipride Roxiam 2 Reserpine Serpasil 2 Rilmazafone 2 Risperidone 2 Ritanserin 2 Rocuronium Zemuron 2 Ropivacaine Naropin 2 Secobarbital (Quinalbarbitone) Seconal 2 Selegiline Eldepryl, Jumex 2

Page 16: Equestrian Canada Drug Classification Scheme

Sertraline Zoloft 2 Snake venoms 2 Somatrem Protropin 2 Somatropin Nutropin 2 Spiclomazine 2 Spiperone 2 Succinylcholine 2 Sulfondiethylmethane 2 Sulfonmethane 2 Sulforidazine Inofal 2 Sulpiride Aiglonyl, Sulpitil 2 Talbutal Lotusate 2 Tandospirone 2 Temazepam Restoril 2 Tetrabenazine Nitoman 2 Tetracaine Pontocaine 2 Tetrazepam Musaril, Myolastin 2 Thebaine 2 Thialbarbital Kemithal 2 Thiamylal Surital 2 Thiethylperazine Torecan 2 Thiopental Pentothal 2 Thioproperazine Majeptil 2 Thioridazine Mellaril 2 Thiothixene Navane 2

Page 17: Equestrian Canada Drug Classification Scheme

Thipropazate Dartal 2 Tiapride Italprid, Luxoben 2 Tiletamine Telazol (with zolazepam) 2 Timiperone Tolopelon 2 Tofisopam Grandazain, Seriel 2 Topiramate Topamax 2 Tramadol Ultram 2 Tranylcypromine Parnate 2 Trazodone Desyrel 2 Tretoquinol Inolin 2 Triazolam Halcion 2 Tribromethanol 2 Tricaine methanesulfonate Finquel, MS-222 2 Trichloroethanol 2 Trichloroethylene Trilene, Trimar 2 Triclofos 2 Trifluomprazine Nortran 2 Trifluoperazine Stelazine 2 Trifluperidol Triperidol 2 Triflupromazine Vetame, Vesprin 2 Trimipramine Surmontil 2 Tubocuarine Metubin, Curare 2 Tybamate Benvil, Nospan 2 Urethane 2 Valnoctamide Nirvanyl 2

Page 18: Equestrian Canada Drug Classification Scheme

Vecuronium Norcuron 2 Venlafaxine Effexor 2 Veralipride Accional, Veralipril 2 Viloxazine Catatrol, Vivalan 2 Vinbarbital Optanox, Speda 2 Zeleplon Sonata 2 Ziprasidone Geodon 2 Zolazepam Telazol (with tiletamine) 2 Zolpidem Ambien 2 Zomepirac Zomax 2 Zopiclone Imovane 2 Zotepine Lodopin 2 Zuclopenthixol Ciatyl, Cesordionl 2 19-Norandrostenediol 3 19-Norandrostenedione 3 4-hydroxytestosterone 3 Acebutolol Sectral 3 Acepromazine Atravet 3 Acetaminophen Tylenol 3 Acetanilide 3 Acetylsalicylic acid Aspirin 3 Aclofenac 3 Almotriptan Axert 3 Alprenolol 3 Ambenonium Mytelase, Myeuran 3

Page 19: Equestrian Canada Drug Classification Scheme

Aminophylline 3 Amiodarone 3 Amitraz Mitaban 3 Amlodipine Norvasc 3 Amlodipine Norvasc 3 Amrinone 3 Amyl nitrate 3 Antipyrine 3 Aprindine 3 Arecholine 3 Atenolol Tenormin 3 Atropine 3 Benazepril Fortekor 3 Bepridil Bepadin 3 Betaxolol Kerlone 3 Bethanidine Esbatal 3 Biperiden Akineton 3 Bisoprolol Zebeta 3 Bitolterol Effectin 3 Bolasterone 3 Boldenone Equipoise 3 Boldione 3 Bretylium Bretylol 3 Brimonidine Alphagan 3 Bromfenac 3

Page 20: Equestrian Canada Drug Classification Scheme

Bromodiphenhydramine 3 Brompheniramine 3 Bufexamac 3 Bumetanide Bumex 3 Butorphanol Torbugesic, Stadol 3 Caffeine 3 Calusterone Methosorb 3 Candesartan Atacand 3 Captopril 3 Carazolol Carbacel 3 Carbachol Lentin 3 Carbamazepine Tegretol 3 Carbinoxamine Clistin 3 Carprofen Rimadyl 3 Carteolol Cartrol 3 Carvedilol Coreg 3 Celecoxib Celebrex 3 Cetirizine Zyrtec 3 Chlorpheniramine Chlor-Tripolon 3 Cimeterol 3 Clemastine Tavist 3 Clenbuterol Ventipulmin 3 Clonidine Catapres 3 Clostebol 3 Cyclandelate Cyclospasmol 3

Page 21: Equestrian Canada Drug Classification Scheme

Cycrimine Pagitane 3 Cyproheptadine Periactin 3 Danazol Danocrine 3 Dehydrochloromethyltestosterone 3 Deracoxib Deramaxx 3 Desoxymethyltestosterone 3 Detomidine Dormosedan 3 Dextropropoxyphene Darvon 3 Diazoxide Proglycem 3 Diclofenac Surpass, Voltaren 3 Diflunisal 3 Digitoxin 3 Digoxin 3 Dihydroergotamine 3 Diltiazem 3 Dimefline 3 Diphenhydramine Benadryl 3 Dipyridamole Persantine 3 Disopyramide 3 Divalproex Depakote 3 Dobutamine Dobutrex 3 Doxazosin 3 Doxylamine Decapryn 3 Dromostanolone 3 Dyphylline 3

Page 22: Equestrian Canada Drug Classification Scheme

Edrophonium Tensilon 3 Eletripan Relpax 3 Eltenac 3 Enalapril (Enalaprilat) Enacard 3 Ephedrine 3 Ergoloid mesylates 3 Ergonovine 3 Ergotamine 3 Erithrityl tetranitrate Cardilate 3 Esmolol Brevibloc 3 Etamiphylline 3 Ethacrynic acid Edecrin 3 Ethosuximide Zarontin 3 Ethylestrenol Maxibolin, Organon 3 Ethylnorepinephrine Bronkephrine 3 Etodolac Lodine 3 Felbamate Felbatol 3 Felodipine 3 Fenbufen Cincopal 3 Fenclozic acid Myalex 3 Fenoldopam Corlopam 3 Fenoprofen Nalfon 3 Fenoterol Berotec 3 Fenspiride Respiride 3 Fentiazac 3

Page 23: Equestrian Canada Drug Classification Scheme

Fexofenadine Allegra 3 Firocoxib Equioxx, Previcox 3 Flecainide 3 Floctafenine 3 Flufenamic acid 3 Fluoxymesterone Halotestin 3 Flupirtine Katadolone 3 Flurbiprofen Froben 3 Formebolone 3 Formoterol Altram 3 Fosinopril (Fosinoprilat) Monopril 3 Fosphenytoin Cerebyx 3 Furazabol 3 Gabapentin Neurontin 3 Glycopyrrolate 3 Guanabenz Wytensin 3 Guanadrel Hylorel 3 Guanethidine Ismelin 3 Heptaminol Corofundol 3 Homatropine Homapin 3 Hydralazine 3 Hydroxyzine Atarax 3 Ibuprofen Advil 3 Ibutilide Corvert 3 Iloprost Ventavis 3

Page 24: Equestrian Canada Drug Classification Scheme

Indomethacin Indocin 3 Ipratropium Atrovent 3 Irbesarten Avapro 3 Isoetharine Bronkosol 3 Isosorbide dinitrate Isordil 3 Isoxicam Maxicam 3 Isradipine DynaCirc 3 Kebuzone 3 Ketorolac Toradol 3 Labetalol Normodyne 3 Lamotrigine Lamictal 3 Levobunolol Betagan 3 Lisinopril Prinivil, Zestril 3 Loratidine Claritin 3 Losartan Hyzaar 3 Mabuterol 3 Mecamylamine Inversine 3 Meclizine Antivert 3 Meclofenamic acid Arquel 3 Medetomidine Domitor 3 Mefenamic acid Ponstel 3 Meloxicam Metacam 3 Mestanolone 3 Mesterolone 3 Metaproterenol Alupent, Metaprel 3

Page 25: Equestrian Canada Drug Classification Scheme

Metenolone 3 Methacholine 3 Methandienone 3 Methandriol Probolic 3 Methandrostenolone Dianabol 3 Methasterone 3 Methdilazine Tacaryl 3 Methixene Trest 3 Methoxamine Vasoxyl 3 Methoxyphenamine Orthoxide 3 Methscopolamine 3 Methsuximide Celontin 3 Methyapyrilene Histadyl 3 Methyl-4-testosterone 3 Methylatropine 3 Methyldienolone 3 Methyldopa Aldomet 3 Methylergonovine 3 Methylnortestosterone 3 Methyltestosterone Metandren 3 Metolazone 3 Metoprolol Lopressor 3 Mexilitine Mexilil 3 Mibolerone 3 Mibrefadil Posicor 3

Page 26: Equestrian Canada Drug Classification Scheme

Midodrine Pro-Amiline 3 Minoxidil Loniten 3 Moexipril (Moexiprilat) Uniretic 3 Muscarine 3 Nadol Corgard 3 Nalbumetone 3 Naloxone Narcan 3 Naltrexone Revia 3 Nandrolone Nandrolin, Laurabolin, Durabolin 3 Naproxen Equiproxen, Naprosyn 3 Naratriptan Amerge 3 Nefopam 3 Neostigmine Prostigmine 3 Nicardipine Cardine 3 Nifedipine Procardia 3 Niflumic acid Nifluril 3 Nimesulide 3 Nimodipine Nemotop 3 Nitroglycerin 3 Norbolethone 3 Norclosterbol 3 Nortestosterone 3 Nylidrine Arlidin 3 Olmesartan Benicar 3 Oxabolone 3

Page 27: Equestrian Canada Drug Classification Scheme

Oxandrolone Anavar 3 Oxaprozin 3 Oxprenolol Trasicor 3 Oxycarbazepine Trieptal 3 Oxymesterone 3 Oxymetholone Androyd, Anadrol 3 Oxyphenbutazone Only class 3 if found without appropriate PBZ concentrations 3 Papaverine Pavagen 3 Paramethadione Paradione 3 Pargyline Eutonyl 3 Penbutolol Levatol 3 Pentaerythritol tetranitrate Duotrate 3 Perindopril Biprel 3 Phenacemide 3 Phenacetin 3 Phenoxybenzamine Dibenzyline 3 Phentolamine Regitine 3 Phenytoin Dilantin 3 Piretanide Arelix, Tauliz 3 Piroxicam Feldene 3 Prazosin Minipress 3 Primidone Mysoline 3 Procainamide 3 Procaine 3 Procaterol Pro Air 3

Page 28: Equestrian Canada Drug Classification Scheme

Procyclidine Kemadrin 3 Promazine 3 Promethazine Phenergan 3 Propafenone 3 Propentophylline Karsivan 3 Propranolol Inderal 3 Prostanazol 3 Protokylol Ventaire 3 Pseudoephedrine 3 Pyridostigmine Mestinon, Regonol 3 Pyrilamine Pyrahist, Antihistamine 3 Quinapril (Quinaprilat) Accupril 3 Quinbolone 3 Quinidine 3 Ramipril (Ramiprilat) Altace 3 Ritodrine Yutopar 3 Rivastigmine Exelon 3 Rizatriptan Maxalt 3 Rofecoxib Vioxx 3 Romifidine Sedivet 3 Salbutamol (Albuterol) Ventolin 3 Salicylamide 3 Salicylate 3 Salmeterol 3 Scopolamine (Hyoscine) Buscopan 3

Page 29: Equestrian Canada Drug Classification Scheme

Sibutramine Meridia 3 Sildenafil Viagra 3 Sotalol Betapace 3 Spirapril (Spiraprilat) Renomax 3 Stanozolol Winstrol 3 Stenbolone 3 Sulindac Clinoril 3 Sumatriptan Imitrex 3 Taladafil Cialis 3 Telmisartin Micardis 3 Tenoxicam Alganex 3 Tepoxalin Zubrin 3 Terazosin Hytrin 3 Terbutaline Bricanyl, Brethine 3 Terfenadine Seldane 3 Testolactone Teslac 3 Testosterone (exogenous) 3 Tetrahydroestrione 3 Theophylline 3 Thiosalicylate 3 Tiaprofenic acid Surgam 3 Timolol Blocardin 3 Tocainide 3 Tolazoline Tolazine 3 Tolmetin Tolectin 3

Page 30: Equestrian Canada Drug Classification Scheme

Trandolapril (Trandolaprilat) Tarka 3 Trenbolone Finaplix 3 Trihexylphenidyl Artane 3 Trimethadione Tridione 3 Trimethaphan Arfonad 3 Tripelennamine 3 Valdecoxib Bextra 3 Valerenic acid 3 Valsartan Diovan 3 Vardenafil Levitra 3 Vedoprofen 3 Verapamil 3 Xylazine Rompun 3 Yohimbine 3 Zolmitriptan Zomig 3 Zonisamide Zonegran 3 2-aminoheptaine Tuamine 4 Acetazolamide 4 Aclomethasone Aclovate 4 Aldosterone Aldocortin 4 Ambroxol 4 Amcinonide Cyclocort 4 Amiloride Moduretic 4 Aminocaproic acid Amicar 4 Aminopyrine 4

Page 31: Equestrian Canada Drug Classification Scheme

Amisometradine Rolictron 4 Anisotropine 4 Azapropazone Rheumox 4 Baclofen Lioresal 4 Beclomethasone Propaderm 4 Bendroflumethiazide Naturetin 4 Betamethasone 4 Bethanechol Urecholine 4 Bromhexine 4 Budesonide Pulmacort 4 Butamben Butesin 4 Calusterone Methosorb 4 Camphor 4 Chlormerodrin Neohydrin 4 Chlorophenesin Maolate 4 Chloroquine Avloclor 4 Chlorothiazide Diuril 4 Chlorthalidone Hydroton 4 Clanobutin 4 Clidinium 4 Clobetasol Temovate 4 Clocotolone Cloderm 4 Clofenamide 4 Colchicine 4 Cortisone 4

Page 32: Equestrian Canada Drug Classification Scheme

Cyclizine Merazine 4 Cyclobenzaprine Flexeril 4 Cyclothiazide 4 Dantrolene Dantrium 4 Dembrexine Sputolysin 4 Deoxycorticosterone Percortin, DOCA 4 Desonite 4 Desoximetasone Topicort 4 Dexamethasone Azium 4 Dextromethorphan 4 Dichlorphenamide Daramide 4 Diflorasone Florone 4 Diflucortolone Flu-Cortinest 4 Dimethylsulfone MSM 4 Dimethylsulfoxide DMSO 4 Diphenoxylate Lomotil 4 Dipyrone 4 Dyclonine 4 Etanercept 4 Ethoheptazine 4 Ethotoin 4 Ethoxyzolamide 4 Flucinolone 4 Fludrocortisone 4 Flumethasone Flucort 4

Page 33: Equestrian Canada Drug Classification Scheme

Flumethiazide 4 Flunarizine 4 Flunisolide 4 Flunixin Banamine 4 Fluocinonide 4 Fluorometholone 4 Flurandrenolide 4 Fluticasone 4 Furosemide Lasix, Salix 4 Halcinonide 4 Halobetasol 4 Hexocyclium 4 Hydrochlorthiazide 4 Hydrocortisone Cortef 4 Hydroflumethiazide 4 Infilximab Remicade 4 Isoflupredone Predef-2X 4 Isometheptene 4 Isopropamide 4 Ketoprofen Anafen 4 Letosteine 4 Medrysone 4 Mellaruide Mercuhydrin 4 Mepenzolate Cantil 4 Mephenesin Tolserol 4

Page 34: Equestrian Canada Drug Classification Scheme

Merbaphen 4 Mercaptomerin Thiomerin 4 Mersalyl 4 Metaxalone 4 Methantheline Banthine 4 Methazolamide Naptazane 4 Methocarbamol Robaxin 4 Methotrexate 4 Methylchlorthiazide 4 Methylprednisolone Medrol 4 Methysergide Sansert 4 Metiamide 4 Metoclopramide Reglan 4 Mometasone Elocon 4 Montelukast Singulair 4 Naepaine Amylsine 4 Naphazoline 4 Olsalazine 4 Orphenadrine Norflex 4 Oxymetazoline Afrin 4 Oxyphencyclimine 4 Paramethasone 4 Pentoxifylline 4 Phenylbutazone 4 Polythiazide 4

Page 35: Equestrian Canada Drug Classification Scheme

Pramoxine 4 Prednisolone 4 Prednisone 4 Probenecid 4 Propantheline 4 Propylhexedrine 4 Spironolactone 4 Tetrahydrozoline 4 Theobromine 4 Thiphenamil 4 Tolmetin 4 Torsemide Demadex 4 Tranexamic acid 4 Triamcinolone Panolog 4 Triamterene 4 Trichlormethiazide Naquasone 4 Tridihexethyl 4 Triprolidine 4 Vedaprofen Quadrisol 4 Xylometazoline 4 Zafirlukast Accolate 4 Zeranol Ralgro 4 Zileuton 4 Acenocoumarol 5 Anisindione 5

Page 36: Equestrian Canada Drug Classification Scheme

Cilostazol 5 Cromolyn 5 Dicoumarol 5 Diphenadione 5 Famotidine 5 Lansoprazole 5 Misoprostol Cytotec 5 Nedocromil Tilade 5 Nizatidine 5 Pantoprazole Protonix, Pantoloc 5 Phenindione 5 Phenprocoumon Liquamar 5 Pirenzapine Gastrozepin 5 Rabeprazole AciPHex, Pariet 5 Warfarin 5