Opposite of dumbbelss, so constipation, urinary retention, tachycardia, bronchorelaxation, loss of stimualation to skeletal muscle, dry eyes/mouth, no sweat
AntiCholinesterase
Direct Muscarinic Agonist
Muscarinic Agonist
Muscarinic Antagonist
Anticholinesterase
Acetylcholinesterase Regenerator
Cholinergic Agonist
Anticholinesterase
Muscarinic Antagonist
Muscarinic Antagonist
Muscarinic Antagonist
Muscarinic Antagonist
Muscarinic Antagonist
Anticholinesterase
Muscarinic Antagonist
Muscarinic Antagonist
Anticholinesterase
Muscarinic Antagonist
Anticholinesterase
Cholinergic Agonist
Ipratropium, Tiotropium
Cocaine, TCA
Calcium, amphetime, ephedrine, tyramine
Cutesies have 1 M&MMAD 2s
Gq
Gi
Gs
Gs
Gq
Gi
Gq
Gi
Gs proteinAdenylcate cyclaseIncreased cAMPProtein Kinase C Activation =
Vd = D/cCL = Rate of elimination/Plasma concentrationCL = (0.7 x Vd) x T1/2LD (loading dose) = Css x VdMD (Maintenance dose) = Css x CL
10.5
600 mg
Stop the infusion for one half life which as we calculated was 10.5 h
20 mg / h
LD will not changeMD will change getting decreased