BIOHETEROCYCLES 2015XVI International Conference on Heterocycles in Bioorganic Chemistry

Campus du SaulcyMetz, France June 8-11, 2015

Plenary LecturesNon Noble Metal Catalysis for Making Precious Molecules Prof. Matthias BELLER (University Rostock, Germany)Heterocycles Derived from Natural Products in Management of Multidrug ResistanceProf. Ahcene BOUMENDJEL (Joseph Fourier University, France)Metal Catalysis for Heteroarene Synthesis Prof. Michael GREANEY (The University of Manchester, United Kingdom)The Discovery and Development of Dolutegravir Dr Brian JOHNS (GlaxoSmithKline, United States)Bronsted Acid and Metal-catalyzed Reactions in the Synthesis of Heterocycles Prof. Esther LETE (University of the Basque Country, Spain)Photoreactive Heterocycles and Natural Product Derivatives Prof. Thomas LINDEL (Technical University of Braunschweig, Germany)Targeting DNA Methylation: a Medicinal Chemistry Approach Prof. Antonello MAI (Sapienza University of Rome, Italy)The Importance of Heterocycles in Agrochemistry: Fungicides as a Case Study Dr Harald WALTER (Syngenta Crop Protection, Switzerland)

Invited LecturersAccess to Heterocycles through Organometallic Catalysis: Study of Silicon-Containing Heterocycles as CDKs InhibitorsProf. Philippe BELMONT (University Paris Descartes, France)Synthetic Explorations in Small-ring Azaheterocyclic Chemistry and Development of Novel Bioactive HeterocyclesProf. Matthias D’HOOGHE (Ghent University, Belgium)TitletobeconfirmedDr Eric DESARBRE (Basilea Pharmaceutica, Switzerland)At the Crossroads of Chemistry and Biology: Inhibiting Protein Kinase CK2 by Heterocyclic Small MoleculesProf. Marc LE BORGNE (University Claude Bernard Lyon 1, France)Utilization of Hypervalent Reagents for the Construction and Functionalization of Heterocyclic MoleculesDr Zoltan NOVAK (Eötvös University, Hungary)New Methods in Thioamide ChemistryDr Mike PORTER (University College London, United Kingdom)Are Generic Drugs Only a Copy_and_Paste Products?Prof. Stanislav RADL (Zentiva, Czech Republic)Synthesis of Novel Alpha7-nAchR Ligands: from an Idea to in Rodent Results for Alzheimer [18F] TEP Imaging Prof. Sylvain ROUTIER (University of Orléans, France)Synthesis of Biorelevant Heterocycles with N-heterocyclic CarbenesProf. Andreas SCHMIDT (Technical University Clausthal, Germany)

www.bioheterocycles2015.eu

Local Organising CommitteeChairmanProf. G. KIRSCH (University of Lorraine, FR)MembersProf. P. CHAIMBAULT (University of Lorraine, FR)Dr C. COMOY (University of Lorraine, FR)Prof. Y. FORT (University of Lorraine, FR)Prof. P. GROS (University of Lorraine, FR)Dr S. HESSE (University of Lorraine, FR)

ScientificCommitteeChairmanProf. J. BERGMAN (Karolinska Institute, SE)MembersProf. M. ÁLVAREZ (Scientifi c Parc of Barcelona, ES)Prof. F. FULOP (University of Szeged, HU)Prof. J. JOULE (The University of Manchester, GB)Prof. M. POTACEK (Masaryk University, CZ)Prof. H. VAN DER PLAS (University of Wageningen, NL)

Important deadlines:Submit your abstract before April 30!

Benefi t from the early bird fee if you register before April 30!

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SYMPOSIUM

A 3.5 days symposium with 8 plenary lectures, 9 invited Lectures, 16 oral communications, a poster session and a scientific exhibition. The symposium will start on Monday June 8, at 09:00.

POSTERS AND ORAL COMMUNICATIONS

Participants wishing to present a poster should submit an abstract via the symposium website, using the abstract submission tool. Submitted abstracts will be peer-reviewed for their acceptance by the Committee. Among the submitted abstracts, 16 oral communications will be selected and the others will have the opportunity to be presented as posters.Deadline for abstract submission: April 30, 2015Website: www.bioheterocycles2015.eu

PRACTICAL INFORMATION

Symposium venue : University of Lorraine, Campus du Saulcy, Île du Saulcy, 57006 Metz - FranceLanguage : The official symposium language is English. No simultaneous translation will be provided.Registration : Please register on-line on the symposium website. The participant registration fee includes:• Admission to all scientific sessions and to the exhibition programme• Abstract book, conference bag and certificate of attendance• Lunches and coffee breaks as per the meeting schedule• Welcome drink on Monday evening• Excursions on Wednesday

REGISTRATION FEES

Profile Earlybirdfeeuntil30/04/2015(EUR) Standardfeeafter30/04/2015(EUR)Accompanying person 75 EUR 90 EURStudent 300 EUR 360 EURAcademic 500 EUR 600 EURIndustry affiliated 650 EUR 780 EUR Activities Price(EUR)June 8 - 18:00 Welcome drink 0 EUR Included in the fee but subject to registrationJune 10 - 16:00 Excursion 1: Walking excursion in Metz 0 EUR (with an English speaking guide). Included in the fee but subject to registration June 10 - 16:00 Excursion 2 - Visit of “Centre Pompidou” 0 EUR Included in the fee but subject to registration June 10 - 19:00 Banquet at the “Abbaye des Prémontrés” 60 EUR

Payment:Payments should preferably be made online while registering for the Symposium on the website www.bioheterocycles2015.euOtherwise, payments can be made by bank transfer (net of all bank costs) to:-Accountn°340-1813781-16(IBANBE72340181378116)-BIC/SWIFTBBRUBEBBBank: ING, Rue des Wallons 2, B-1348 Louvain-la-Neuve, BelgiumParticipants from France can proceed with a transfer to:-Accountn°09350000672(IBANFR7630056009350935000067272)-BIC/SWIFTCCFRFRPPBank: HSBC France, CAE Paris Rive Gauche - 107 bd St. Germain, F-75006 Paris, FrancePlease mention «Bioheterocycles 2015» and your references in the transfer.

Cancellations:Substitutions may be made at any time, by advising the Symposium Secretariat by written notice of any change of name.Cancellations should be sent by written notice to the Symposium Secretariat and cancellation fees will apply as follows:• Cancellation notice prior to 60 days before the start of the event: registration fees will be refunded, less €125,00 processing

charges (these charges are reduced to 40% of the payment in case the registration fee is less than €125,00)• Cancellation notice between 60 days and 30 days prior to the start of the event: 50% of the registration fees will be due, with a

minimum of €125,00 (except when the registration fee is less than €125,00)• Cancellation notice less than 30 days before the start of the event: no cancellation refund can be given

ACCOMMODATION

Options have been taken on low budget studios in the Aparthotel Residhome (30 min walking distance), partner of the University of Metz. (10 rue Lafayette - 57000 Metz) Price: 59 € per night for 1 or 2 persons, breakfast: 10 € per person, tax: 0.95 € per person.Other hotels are also available on the Accor website. Check the accommodation page on www.bioheterocycles2015.eu for more information.

SYMPOSIUM SECRETARIAT

LD Organisation sprl | Scientific Conference ProducersRue Michel de Ghelderode 33/2 |B-1348 Louvain-La-NeuvreTel: +32 10 454777 | Fax: +32 10 459719Email: secretariat@ldorganisation.com | Web: www.bioheterocycles2015.eu

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